Synthesis of Substituted Pyrido-oxazine through Tandem SN2 and SNAr Reaction
نویسندگان
چکیده
منابع مشابه
A one-pot asymmetric organocatalytic tandem reaction for the synthesis of oxazine derivatives.
An easy one-pot tandem reaction catalyzed by a chiral secondary amine for the synthesis of optically active oxazine derivatives has been performed and the corresponding substituted benzo[d]pyrido[2,1-b][1,3]oxazine derivatives were afforded in generally high yields (up to 99%) and excellent enantioselectivities (up to >99%).
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ژورنال
عنوان ژورنال: SynOpen
سال: 2018
ISSN: 2509-9396
DOI: 10.1055/s-0036-1591960